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Tesofensine (with metoprolol) tesofensine is a presynaptic uptake inhibitor of noradrenaline, dopamine and serotonin. · tesofensine is a compound originally developed for the treatment of neurological diseases such as alzheimers … · abstract tesofensine (te) is a novel triple monoamine re-uptake inhibitor inducing a potent inhibition of the re-uptake process in … · tesofensine tesofensine is an inhibitor of neuronal reuptake of dopamine, noradrenaline, and serotonin. Tesofensine tesofensine is a dopamine, serotonin, and noradrenaline (triple) reuptake inhibitor originally developed by neurosearch … There has been …